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Fosaprepitant dimeglumine

CAS No. 265121-04-8

Fosaprepitant dimeglumine ( MK 0517 )

产品货号. M13812 CAS No. 265121-04-8

Fosaprepitant dimeglumine(MK-0517) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting.

纯度: >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
5MG ¥365 有现货
10MG ¥494 有现货
25MG ¥996 有现货
50MG ¥1806 有现货
100MG ¥2989 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Fosaprepitant dimeglumine
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Fosaprepitant dimeglumine(MK-0517) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting.
  • 产品描述
    Fosaprepitant dimeglumine(MK-0517) is a neurokinin-1 receptor antagonist for the prevention of chemotherapy-induced nausea and vomiting.
  • 同义词
    MK 0517
  • 通路
    GPCR/G Protein
  • 靶点
    Neurokinin Receptor
  • 受体
    NK1
  • 研究领域
    Neurological Disease
  • 适应症
    ——

化学信息

  • CAS Number
    265121-04-8
  • 分子量
    1004.83
  • 分子式
    C37H56F7N6O16P
  • 纯度
    >98%(HPLC)
  • 溶解度
    Water: 135 mg/mL (134.35 mM); DMSO: 201 mg/mL (200.03 mM)
  • SMILES
    C[C@H](C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)O[C@@H]2[C@@H](N(CCO2)CC3=NC(=O)N(N3)P(=O)(O)O)C4=CC=C(C=C4)F.CNC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O.CNC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.Navari RM. Expert Opin Investig Drugs, 2007, 16(12), 1977-1985.
产品手册
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